发明名称 |
UREA ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS |
摘要 |
The present invention provides novel pyridyl or phenyl ureas and analogues thereof, which are selective inhibitors of the human P2Y<SUB>1 </SUB>receptor. The invention also provides for various pharmaceutical compositions of the same and methods for treating diseases responsive to modulation of P2Y<SUB>1 </SUB>receptor activity.
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申请公布号 |
US2008280905(A1) |
申请公布日期 |
2008.11.13 |
申请号 |
US20080117005 |
申请日期 |
2008.05.08 |
申请人 |
BRISTOL MYERS SQUIBB COMPANY |
发明人 |
CHAO HANNGUANG J.;TUERDI HUJI;HERPIN TIMOTHY F.;ROBERGE JAQUES YVES;LIU YALEI;LAWRENCE R. MICHAEL;REHFUSS ROBERT P.;CLARK CHARLES G.;QIAO JENNIFER X.;GUNGOR TIMUR;LAM PATRICK Y. S.;WANG TAMMY;RUEL REJEAN;L'HEUREUX ALEXANDRE;THIBEAULT CARL;BOUTHILLIER GILLES;SCHNUR DORA M. |
分类号 |
A61K31/5377;A61K31/4412;A61K31/4439;A61K31/444;A61K31/4545;A61K31/4709;A61K31/4725;A61K31/496;A61K31/501;A61P7/00;A61P9/00;C07C275/30;C07C275/32;C07D213/40;C07D213/72;C07D213/75;C07D213/89;C07D231/40;C07D231/50;C07D237/22;C07D333/36;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07F7/18 |
主分类号 |
A61K31/5377 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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