发明名称 UREA ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS
摘要 The present invention provides novel pyridyl or phenyl ureas and analogues thereof, which are selective inhibitors of the human P2Y<SUB>1 </SUB>receptor. The invention also provides for various pharmaceutical compositions of the same and methods for treating diseases responsive to modulation of P2Y<SUB>1 </SUB>receptor activity.
申请公布号 US2008280905(A1) 申请公布日期 2008.11.13
申请号 US20080117005 申请日期 2008.05.08
申请人 BRISTOL MYERS SQUIBB COMPANY 发明人 CHAO HANNGUANG J.;TUERDI HUJI;HERPIN TIMOTHY F.;ROBERGE JAQUES YVES;LIU YALEI;LAWRENCE R. MICHAEL;REHFUSS ROBERT P.;CLARK CHARLES G.;QIAO JENNIFER X.;GUNGOR TIMUR;LAM PATRICK Y. S.;WANG TAMMY;RUEL REJEAN;L'HEUREUX ALEXANDRE;THIBEAULT CARL;BOUTHILLIER GILLES;SCHNUR DORA M.
分类号 A61K31/5377;A61K31/4412;A61K31/4439;A61K31/444;A61K31/4545;A61K31/4709;A61K31/4725;A61K31/496;A61K31/501;A61P7/00;A61P9/00;C07C275/30;C07C275/32;C07D213/40;C07D213/72;C07D213/75;C07D213/89;C07D231/40;C07D231/50;C07D237/22;C07D333/36;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07F7/18 主分类号 A61K31/5377
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