发明名称 |
CARBONIC ANHYDRASE INHIBITORS DERIVATIVES |
摘要 |
Nitroderivatives of dorzolamide and brinzolamide having improved pharmacological activity and enhanced tolerability are described. They can be employed for the treatment of glaucoma, ocular hypertension, age-related macular degeneration, diabetic macular edema, diabetic retinopathy, hypertensive retinopathy and retinal vasculopathies. |
申请公布号 |
WO2008075155(A3) |
申请公布日期 |
2008.11.06 |
申请号 |
WO2007IB03856 |
申请日期 |
2007.12.03 |
申请人 |
NICOX S.A.;PFIZER INC.;BENEDINI, FRANCESCA;BIONDI, STEFANO;ONGINI, ENNIO |
发明人 |
BENEDINI, FRANCESCA;BIONDI, STEFANO;ONGINI, ENNIO |
分类号 |
C07D495/04;A61K31/38;A61K31/542;C07D513/04 |
主分类号 |
C07D495/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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