| 发明名称 |
Semisynthesis process for the preparation of 10-deacetyl-N-debenzoyl-paclitaxel |
| 摘要 |
A process is provided for the preparation of 10-deacetyl-N-debenzoyl-paclitaxel (I) a synthon useful for the preparation of taxanes with antitumour activity, and intermediates for the preparation thereof. Also described is a process for the preparation of Docetaxel starting from the compound of formula (I).
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| 申请公布号 |
US7446126(B2) |
申请公布日期 |
2008.11.04 |
| 申请号 |
US20050244171 |
申请日期 |
2005.10.06 |
| 申请人 |
INDENA S.P.A. |
发明人 |
GABETTA BRUNO;GAMBINI ANDREA;BOMBARDELLI EZIO;FONTANA GABRIELE |
| 分类号 |
A01N43/02;A61K31/335;C07D305/00;C07D407/00;C07D493/00 |
主分类号 |
A01N43/02 |
| 代理机构 |
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| 主权项 |
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