发明名称 POLYMORPHIC FORMS OF RIMONABANT BASE AND PROCESSES FOR PREPARATION THEREOF
摘要 The present invention provides process for crystalline forms of Rimonabant base, including processes that prepare crystalline forms of Rimonabant base. Also provided is a crystalline Rimonabant base form I having a substantially reduced residual solvent content, including processes that prepare such crystalline Rimonabant form I. These crystalline forms of Rimonabant base may be in a pharmaceutical compositions further comprising at least one pharmaceutically acceptable excipient.
申请公布号 WO2008088900(A3) 申请公布日期 2008.10.30
申请号 WO2008US00726 申请日期 2008.01.18
申请人 TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARMACEUTICALS USA, INC.;RAFILOVICH, MICHAL;LIFSHITZ-LIRON, REVITAL;ARONHIME, JUDITH;KALUJNY, MARINA;LANCRY, ELI;SHMUELY, YARON 发明人 RAFILOVICH, MICHAL;LIFSHITZ-LIRON, REVITAL;ARONHIME, JUDITH;KALUJNY, MARINA;LANCRY, ELI;SHMUELY, YARON
分类号 C07D231/14;A61K31/415;A61P25/00 主分类号 C07D231/14
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