发明名称 |
A NEW PROCESS FOR THE MANUFACTURING OF THE COMPOUND 2-HYDROXY-3-[5-(MORPHOLIN-4-YLMETHYL)PYRIDIN-2-YL]1H-INDOLE-5-CARBONITRILE 701 |
摘要 |
The present invention relates to a new process for the manufacture of the compound 2-hydroxy-3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]1H-indole-5-carb onitrile as a free base and pharmaceutically acceptable salts thereof, parti cularly the 2-hydroxy-3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]1H-indole-5-ca rbonitrile citrate, and to new intermediates prepared in said process suitab le for large scale manufacturing of said compound.
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申请公布号 |
CA2684347(A1) |
申请公布日期 |
2008.10.30 |
申请号 |
CA20082684347 |
申请日期 |
2008.04.17 |
申请人 |
ASTRAZENECA AB |
发明人 |
THIERING, SWANTJE;RYBERG, PER;JANSSON, ANNETTE;HEDBERG, MARTIN;DELISSER, VERN;RADEVIK, ANDREAS |
分类号 |
C07D401/04;A61K31/5355;C07D213/38 |
主分类号 |
C07D401/04 |
代理机构 |
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地址 |
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