发明名称 SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE
摘要 This invention comprises the novel compounds of formula (I) wherein R, RRX and Y have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
申请公布号 EA010652(B1) 申请公布日期 2008.10.30
申请号 EA20070000138 申请日期 2005.07.25
申请人 JANSSEN PHARMACEUTICA N.V. 发明人 VERDONCK MARC, GUSTAAF, CELINE;ANGIBAUD PATRICK, RENE;ROUX BRUNO;PILATTE ISABELLE, NOELLE, CONSTANCE;TEN HOLTE PETER;ARTS JANINE;VAN EMELEIN KRISTOF
分类号 C07D401/14;A61K31/506;A61P35/00;C07D405/14;C07D409/14 主分类号 C07D401/14
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