| 发明名称 |
DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONISTS |
| 摘要 |
A compound of the formula (I) wherein the variables X<SUB>1 </SUB>to X<SUB>10</SUB>, R<SUP>1 </SUP>to R<SUP>7 </SUP>including R<SUP>3'</SUP>, E, v, y, z. A and B are as described, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixtures thereof, useful for the treatment, prevention or amelioration of obesity and Related Diseases is disclosed.
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| 申请公布号 |
US2008269296(A1) |
申请公布日期 |
2008.10.30 |
| 申请号 |
US20080052972 |
申请日期 |
2008.03.21 |
| 申请人 |
BLANCO-PILLADO MARIA-JESUS;CHAPPELL MARK DONALD;DE LA TORRE MARTA GARCIA;DIAZ BUEZO NURIA;FRITZ JAMES ERWIN;HOLLOWAY WILLIAM GLEN;MATT JAMES EDWARD;MITCH CHARLES HOWARD;PEDREGAL-TERCERO CONCEPCION;QUIMBY STEVEN JAMES;SIEGEL MILES GOODMAN;SMITH DANA RAE;STUCKY RUSSELL DEAN;TAKEUCHI KUMIKO;THOMAS ELIZABETH MARIE;WOLFE CHAD NOLAN |
发明人 |
BLANCO-PILLADO MARIA-JESUS;CHAPPELL MARK DONALD;DE LA TORRE MARTA GARCIA;DIAZ BUEZO NURIA;FRITZ JAMES ERWIN;HOLLOWAY WILLIAM GLEN;MATT JAMES EDWARD;MITCH CHARLES HOWARD;PEDREGAL-TERCERO CONCEPCION;QUIMBY STEVEN JAMES;SIEGEL MILES GOODMAN;SMITH DANA RAE;STUCKY RUSSELL DEAN;TAKEUCHI KUMIKO;THOMAS ELIZABETH MARIE;WOLFE CHAD NOLAN |
| 分类号 |
A61K31/4433;A61P3/04;A61P25/32;C07C235/46;C07D213/38;C07D213/64;C07D213/643;C07D213/78;C07D213/81;C07D213/82;C07D217/04;C07D237/24;C07D241/24;C07D307/14;C07D333/20;C07D401/06;C07D401/12;C07D401/14;C07D405/12;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07D417/14 |
主分类号 |
A61K31/4433 |
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