发明名称 [2, 6] NAPHTHYRIDINES USEFUL AS PROTEIN KINASE INHIBITORS
摘要 <p>The present invention provides a compound of formula I: (formula I) said compound is inhibitor of selective subset of kinases belonging to the AGC or calmodulin kinase family, such as for example MARK1/2/3, PKD-1/2/3, PKN-1/2, CDK-9, CaMKII, ROCK-I/II, inhibitors of histone deacetylase (HDAC) phosphorylation, or inhibitors of other kinases. Finally, the present invention also provides a pharmaceutical composition.</p>
申请公布号 WO2008122615(A1) 申请公布日期 2008.10.16
申请号 WO2008EP54105 申请日期 2008.04.04
申请人 NOVARTIS AG;DOBLER, MARKUS ROLF;JEWELL, CHARLES FRANCIS JR;MEREDITH, ERIK;MONOVICH, LAUREN G.;SISKA, SARAH;VON MATT, ANETTE;VAN EIS, MAURICE;YOON, TAEYOUNG;GAUL, CHRISTOPH;CAPPARELLI, MICHAEL PAUL 发明人 DOBLER, MARKUS ROLF;JEWELL, CHARLES FRANCIS JR;MEREDITH, ERIK;MONOVICH, LAUREN G.;SISKA, SARAH;VON MATT, ANETTE;VAN EIS, MAURICE;YOON, TAEYOUNG;GAUL, CHRISTOPH;CAPPARELLI, MICHAEL PAUL
分类号 C07D471/04;A61K31/4375;A61P35/00;C07D519/00 主分类号 C07D471/04
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