发明名称 DEVELOPMENT OF MOLECULAR IMAGING PROBES FOR CARBONIC ANHYDRASE-IX USING CLICK CHEMISTRY
摘要 The present application discloses methods for identifying inhibitors with high binding-affinity for the carbonic anhydrase-IX (CA-IX) enzyme using cl ick chemistry and uses the candidates thereof as positron emission tomograph y (PET) imaging agents.
申请公布号 CA2683434(A1) 申请公布日期 2008.10.16
申请号 CA20082683434 申请日期 2008.04.07
申请人 SIEMENS MEDICAL SOLUTIONS USA, INC. 发明人 WALSH, JOSEPH C.;KASI, DHANALAKSHMI;XIA, CHUNFANG;DUCLOS, BRIAN A.;GANGADHARMATH, UMESH B.;WANG, BING;MOCHARLA, VANI;GAO, ZHIYONG;LIANG, QIANWA;SCOTT, PETER J. H.;PADGETT, HENRY CLIFTON;KARIMI, FARHAD;ZHAO, TIEMING;ZHANG, WEI;COLLIER, THOMAS LEE;CHEN, GANG;CHEN, KAI;KOLB, HARTMUTH C
分类号 C07D249/04;A61K31/4192;A61P35/00;C07D249/06;C07D401/04;C07D401/12;C07D403/04;C07D403/12;C07D405/04;C07D405/12;C07D409/12;C07D417/04;C07D417/12;C07D417/14;G01N33/532 主分类号 C07D249/04
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