发明名称 |
NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS |
摘要 |
Compounds of formula I, wherein R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>a</SUP>, X, X<SUP>1</SUP>, and Y are as defined herein or pharmaceutically acceptable salts thereof, inhibit HIV-1 reverse transcriptase and afford a method for prevention and treatment of HIV-1 infections and the treatment of AIDS and/or ARC. The present invention also relates to compositions containing compounds of formula 1 useful for the prevention and treatment of HIV-1 infections and the treatment of AIDS and/or ARC. |
申请公布号 |
WO2008122534(A2) |
申请公布日期 |
2008.10.16 |
申请号 |
WO2008EP53806 |
申请日期 |
2008.03.31 |
申请人 |
F. HOFFMANN-LA ROCHE AG;BILLEDEAU, ROLAND J.;PALMER, WYLIE SOLANG;SWEENEY, ZACHARY KEVIN;WU, JEFFREY |
发明人 |
BILLEDEAU, ROLAND J.;PALMER, WYLIE SOLANG;SWEENEY, ZACHARY KEVIN;WU, JEFFREY |
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