发明名称 PYRIMIDINE HYDRAZIDE COMPOUNDS AS PGDS INHIBITORS
摘要 <p>This invention is directed to a compound wherein R&lt;SUP&gt;1,&lt;/SUP&gt; R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, R&lt;SUP&gt;4&lt;/SUP&gt; and L&lt;SUP&gt;1&lt;/SUP&gt; are as defined herein, a pharmaceutical composition comprising the compound, and the use of the compound to treat allergic and/or inflammatory disorders, particularly disorders such as allergic rhinitis, asthma and/or chronic obstructive pulmonary disease (COPD).</p>
申请公布号 WO2008121670(A1) 申请公布日期 2008.10.09
申请号 WO2008US58347 申请日期 2008.03.27
申请人 SANOFI-AVENTIS;ALDOUS, SUZANNE, C.;FENNIE, MICHAEL, W.;JIANG, JOHN, Z.;JOHN, STANLY;MU, LAN;PEDGRIFT, BRIAN;PRIBISH, JAMES, R.;RAUCKMAN, BARBARA;SABOL, JEFFREY, S.;STOKLOSA, GRZEGORZ, T.;THURAIRATNAM, SUKANTHINI;VANDEUSEN, CHRISTOPHER, L. 发明人 ALDOUS, SUZANNE, C.;FENNIE, MICHAEL, W.;JIANG, JOHN, Z.;JOHN, STANLY;MU, LAN;PEDGRIFT, BRIAN;PRIBISH, JAMES, R.;RAUCKMAN, BARBARA;SABOL, JEFFREY, S.;STOKLOSA, GRZEGORZ, T.;THURAIRATNAM, SUKANTHINI;VANDEUSEN, CHRISTOPHER, L.
分类号 C07D239/28;A61K31/506;A61P29/00;C07D403/12;C07D403/14;C07D413/12;C07D417/14 主分类号 C07D239/28
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