发明名称 GLUCOPYRANOSYLOXYPYRAZOLE DERIVATIVES, MEDICINAL COMPOSITIONS CONTAINING THE SAME AND INTERMEDIATES IN THE PRODUCTION THEREOF
摘要 The present invention relates to glucopyranosyloxy- pyrazole derivatives represented by the general formula: wherein R1 represents a hydrogen atom or a lower alkyl group; one of Q1 and T1 represents a group represented by the general formula: while the other represents a lower alkyl group or a halo ( lower alkyl) group; and R2 represents a hydrogen atom, a lower alkyl group, a lower alkoxy group, a lower alkylthio group, a halo(lower alkyl) group or a halogen atom, or pharmaceutically acceptable salts thereof, which have an inhibitory activity in human SGLT2 and are useful as agents for the prevention or treatment of diabetes, diabetic complications or obesity, and to pharmaceutical compositions comprising the same and intermediates thereof.
申请公布号 CA2382480(C) 申请公布日期 2008.09.30
申请号 CA20002382480 申请日期 2000.08.24
申请人 KISSEI PHARMACEUTICAL CO. LTD. 发明人 NISHIMURA, TOSHIHIRO;FUJIKURA, HIDEKI;ISAJI, MASAYUKI;FUJIOKA, MINORU;HIRATOCHI, MASAHIRO;KATSUNO, KENJI;IYOBE, AKIRA
分类号 C07H17/02;A61K31/7056;A61P3/04;A61P3/10;C07D231/20 主分类号 C07H17/02
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