发明名称 POLYMORPH B OF A KNOWN THIOPHENECARBOXYLIC DODECAHYDROCYCLOPENTA [A]PHENANTHRENYL ESTER
摘要 POLYMORPHIC CRYSTAL FORMS OF 3-METHYLTHIOPHENE-2-CARBOXYLIC ACID @(6S, 9R, 10S, 11S, 13S, 16R, 17R)-9-CHOLORO-6-FLUORO-11-HYDROXY-@17-METHOXYCARBONYL-10, 13, 16,-TRIMETHYL-3-OXO-6, 7, 8, 9, 10,11, 12, 13, 14, 15, 16, 17-DODECAHYDRO-3H-CYCLOPENTA[A]PHENANTHREN-17-YL ESTER. THE CRYSTAL FORMS POSSESS ANTI-INFLAMMATORY ACTIVITY AND HAVE VERY GOOD STABILITY. METHODS FOR PREPARING THE CRYSTAL FORMS ARE ALSO DESCRIBED.
申请公布号 MY136407(A) 申请公布日期 2008.09.30
申请号 MYPI20032832 申请日期 2003.07.28
申请人 NOVARTIS AG 发明人 GUIDO JORDINE;MICHAEL MUTZ
分类号 A61P11/00;C07J33/00 主分类号 A61P11/00
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