发明名称 |
PROCESS FOR SYNTHESIZING ASPARTIC AND GLUTAMIC ACID DERIVATIVES ESPECIALLY USEFUL AS INTERMEDIATES IN THE MANUFACTURE OF A CASPASE INHIBITOR |
摘要 |
The invention relates to novel diazoketone derivatives. The invention also relates to processes for homologation of these diazoketone derivatives. The processes are useful for preparing compounds that are caspase inhibitors.
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申请公布号 |
US2008227976(A1) |
申请公布日期 |
2008.09.18 |
申请号 |
US20080030833 |
申请日期 |
2008.02.13 |
申请人 |
VERTEX PHARMACEUTICALS INCORPORATEAD |
发明人 |
MORTIMORE MICHAEL;PHILPS OLIVER;STUDLEY JOHN |
分类号 |
C07D243/10;C07F7/18;C07C227/32;C07C229/24;C07C229/28;C07C245/00;C07C245/04;C07C245/18;C07D209/42 |
主分类号 |
C07D243/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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