发明名称 PROCESS FOR SYNTHESIZING ASPARTIC AND GLUTAMIC ACID DERIVATIVES ESPECIALLY USEFUL AS INTERMEDIATES IN THE MANUFACTURE OF A CASPASE INHIBITOR
摘要 The invention relates to novel diazoketone derivatives. The invention also relates to processes for homologation of these diazoketone derivatives. The processes are useful for preparing compounds that are caspase inhibitors.
申请公布号 US2008227976(A1) 申请公布日期 2008.09.18
申请号 US20080030833 申请日期 2008.02.13
申请人 VERTEX PHARMACEUTICALS INCORPORATEAD 发明人 MORTIMORE MICHAEL;PHILPS OLIVER;STUDLEY JOHN
分类号 C07D243/10;C07F7/18;C07C227/32;C07C229/24;C07C229/28;C07C245/00;C07C245/04;C07C245/18;C07D209/42 主分类号 C07D243/10
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