| 发明名称 |
5-SULPHANYL-4H-1,2,4-TRIAZOLE DERIVATIVE AND THEIR USE AS MEDICINAL AGENTS |
| 摘要 |
FIELD: chemistry. ^ SUBSTANCE: new 5-sulphanyl-4H-1,2,4-triazole derivatives of general formula I (meaning of radicals R1-R3 are indicated in the description of the invention), methods of their preparation by liquid-phase parallel synthesis and pharmaceutical composition are claimed. ^ EFFECT: claimed compounds display high affinity to some subtypes of somostatin receptors of the SST2 and SST5 subtypes and possibility of their usage for treatment of pathological states or diseases involving one or more of the given somostatin receptors ^ 9 cl, 708 ex |
| 申请公布号 |
RU2367655(C2) |
申请公布日期 |
2009.09.20 |
| 申请号 |
RU20040119406 |
申请日期 |
2002.11.27 |
| 申请人 |
SOS'ETE DE KONSEJ DE RESHERSH EH D`APPLIKAS'ON S'ENTIFIK (S.K.R.A.S.) |
发明人 |
GAL'SERA KONTUR MARI-ODIL';SIDJU AL'BAN;RUBER P'ER;TJUR'O KRISTOF |
| 分类号 |
A61K31/4196;A61K31/433;A61K31/4439;A61K31/454;A61K31/4725;A61K31/498;A61P1/00;A61P1/04;A61P1/12;A61P1/16;A61P1/18;A61P3/04;A61P3/10;A61P5/00;A61P5/02;A61P5/16;A61P5/48;A61P9/02;A61P11/00;A61P13/12;A61P15/00;A61P17/00;A61P17/06;A61P19/00;A61P19/10;A61P25/00;A61P25/08;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P27/02;A61P29/00;A61P35/00;A61P35/02;A61P43/00;C07D249/12;C07D401/04;C07D401/12;C07D401/14;C07D403/04;C07D403/12;C07D403/14;C07D405/04;C07D405/12;C07D409/04;C07D409/14;C07D417/04;C07D471/04 |
主分类号 |
A61K31/4196 |
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