发明名称 SALTS, PRODRUGS AND POLYMORPHS OF FAB I INHIBITORS
摘要 Salts of compounds according to formula (I) wherein the X is selected from the group consisting of H<SUB>2</SUB>SO<SUB>4</SUB>, HSO<SUB>3</SUB>R', HSO<SUB>3</SUB>Ar, H<SUB>3</SUB>PO<SUB>4</SUB>, HCl, HBr, CF<SUB>3</SUB>CO<SUB>2</SUB>H and CCl<SUB>3</SUB>CO<SUB>2</SUB>H. The preferred salt being the p-toluene sulfonate. These compounds and their pharmaceutical composition are useful as Fabl inhibitors for treating bacterial infections.
申请公布号 WO2008098374(A1) 申请公布日期 2008.08.21
申请号 WO2008CA00300 申请日期 2008.02.15
申请人 AFFINIUM PHARMACEUTICALS, INC.;PAULS, HENRY;RAMNAUTH, JAILALL 发明人 PAULS, HENRY;RAMNAUTH, JAILALL
分类号 C07D471/04;A61K31/4375;A61L2/16;A61P31/04 主分类号 C07D471/04
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