发明名称 |
CRYSTALLINE ACID-ADDITION SALT OF CEFDINIR AND CEFDINIR PRODUCTION METHOD USING THE SAME |
摘要 |
PROBLEM TO BE SOLVED: To provide a crystalline acid-addition salt from cefdinir; to provide a production method of the acid-addition salt; and to provide a cefdinir production method using the acid-addition salt. SOLUTION: High purity cefdinir can be produced by a method comprising a step of preparing a crystalline cefdinir salt by reacting a cefdinir intermediate with a mixture acid of formic acid-sulfuric acid or formic acid-methane sulfonic acid and a step of reacting the resultant crystalline salt with a base in a solvent. COPYRIGHT: (C)2008,JPO&INPIT
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申请公布号 |
JP2008189688(A) |
申请公布日期 |
2008.08.21 |
申请号 |
JP20080099293 |
申请日期 |
2008.04.07 |
申请人 |
HANMI PHARM CO LTD |
发明人 |
GUWAN-SUN RII;CHANG YOUNG KIL;KIM HONG SEON;PARK CHUL-HYUN;PARK GHA-SEUNG;KIM CHEOL-KYUNG |
分类号 |
C07D501/22;C07B61/00;C07D501/00;C07D501/14 |
主分类号 |
C07D501/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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