发明名称 |
A 2-F LUOROBENZOATE SALT AND A 2, 6-DIF LUOROBENZOATE SALT OF N-{5-CHLORO-2- [ ( (2S) -3-{ [1- (4-CHLOROBENZYL)PIPERIDIN-4- YL ] AMINO } - 2 - HYDROXY- 2 -ME T HYLPR OPYL ) OXY] - 4 - HYDROXYPHENYL } ACETAMIDE |
摘要 |
<p>The invention provides a 2-fluorobenzoate salt and a 2,6-difluorobenzoate salt of N-{5-chloro-2-[((2S)-3-{[1-(4-chlorobenzyl)piperidin-4-yl]amino}-2-hydroxy-2-methylpropyl)oxy]-4-hydroxyphenyl}acetamide or a solvate and polymorhpic forms thereof, pharmaceutical compositions containing the salts or solvates and use thereof in therapy.</p> |
申请公布号 |
WO2008100202(A1) |
申请公布日期 |
2008.08.21 |
申请号 |
WO2008SE00118 |
申请日期 |
2008.02.13 |
申请人 |
ASTRAZENECA AB;GIOVANNINI, JULIEN;JOSEFSSON, BO-GOERAN;MENSONIDES-HARSEMA, MARGUERITE;SCHULZ, HAAKAN |
发明人 |
GIOVANNINI, JULIEN;JOSEFSSON, BO-GOERAN;MENSONIDES-HARSEMA, MARGUERITE;SCHULZ, HAAKAN |
分类号 |
C07D211/58;A61K9/72;A61K31/4468;A61P11/00;A61P11/06 |
主分类号 |
C07D211/58 |
代理机构 |
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代理人 |
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地址 |
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