发明名称 1,1-DIOXO-1-THIA-5,10-DIAZADIBENZOCYCLOHEPTENES USEFUL AS HEPATITIS C VIRUS INHIBITORS
摘要 <p>Inhibitors of HCV replication of formula (I) the stereoisomers, prodrugs, tautomers, racemics, salts, hydrates or solvates thereof wherein R&lt;SUP&gt;1a&lt;/SUP&gt;; R&lt;SUP&gt;1b&lt;/SUP&gt; R&lt;SUP&gt;2&lt;/SUP&gt;; R&lt;SUP&gt;3&lt;/SUP&gt;; R&lt;SUP&gt;4a&lt;/SUP&gt; and R&lt;SUP&gt;4b&lt;/SUP&gt; have the meaning defined in the claims. The present invention also relates to processes for preparing said compounds, pharmaceutical compositions containing them and their use in HCV therapy.</p>
申请公布号 WO2008099020(A1) 申请公布日期 2008.08.21
申请号 WO2008EP51903 申请日期 2008.02.15
申请人 TIBOTEC PHARMACEUTICALS LTD.;RABOISSON, PIERRE JEAN-MARIE BERNARD;VANDYCK, KOEN;NYANGUILE, ORIGENE;MC GOWAN, DAVID CRAIG;VENDEVILLE, SANDRINE MARIE HELENE;AMSSOMS, KATIE INGRID EDUARD;BOUTTON, CARLO WILLY MAURICE;LORY, PEDRO MIGUEL JALES;HU, LILI;VAN DEN BROECK, WALTER MARCEL MATHILDE;CUMMINGS, MAXWELL DAVID;ROMBAUTS, KLARA;LAST, STEFAAN JULIEN;TAHRI, ABDELLAH 发明人 RABOISSON, PIERRE JEAN-MARIE BERNARD;VANDYCK, KOEN;NYANGUILE, ORIGENE;MC GOWAN, DAVID CRAIG;VENDEVILLE, SANDRINE MARIE HELENE;AMSSOMS, KATIE INGRID EDUARD;BOUTTON, CARLO WILLY MAURICE;LORY, PEDRO MIGUEL JALES;HU, LILI;VAN DEN BROECK, WALTER MARCEL MATHILDE;CUMMINGS, MAXWELL DAVID;ROMBAUTS, KLARA;LAST, STEFAAN JULIEN;TAHRI, ABDELLAH
分类号 C07D495/04;A61K31/55;A61P31/00 主分类号 C07D495/04
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