PLATINUM ANALOGS WITH BIS-NITRILE-CONTAINING LIGANDS
摘要
<p>Disclosed herein are novel platinum-based analogs possessing two nitrile substituent groups (bis-nitrile) covalently-bonded to the platinum. Also disclosed herein are the reaction schemes for the synthesis of said platinum complexes, as well as quantitative in vitro IC50 data.</p>
申请公布号
WO2008100301(A1)
申请公布日期
2008.08.21
申请号
WO2007US22893
申请日期
2007.10.30
申请人
BIONUMERIK PHARMACEUTICALS, INC.;CHEN, XINGHAI;PETLURU, PAVANKUMAR, N.V.;HUANG, QIULI;NARKUNAN, KESAVARAM;HAUSHEER, FREDERICK, H.
发明人
CHEN, XINGHAI;PETLURU, PAVANKUMAR, N.V.;HUANG, QIULI;NARKUNAN, KESAVARAM;HAUSHEER, FREDERICK, H.