发明名称 HCV INHIBITING MACROCYCLIC PHOSPHONATES AND AMIDOPHOSPHATES
摘要 <p>Inhibitors of HCV replication of Formula (I) the /V-oxides, salts, and stcreochcmically isomeric forms thereof; pharmaceutical compositions containing compounds (1) and processes for preparin compounds (I). The side chain R&lt;SUP&gt;2&lt;/SUP&gt; is an amidophosphate or a phosphonate group and X, R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, E and n are as defined in the application.</p>
申请公布号 WO2008096002(A1) 申请公布日期 2008.08.14
申请号 WO2008EP51558 申请日期 2008.02.08
申请人 TIBOTEC PHARMACEUTICALS LTD.;MEDIVIR AB;ANTONOV, DMITRY;NILSSON, KARL, MAGNUS;RABOISSON, PIERRE JEAN-MARIE BERNARD;ROSENQUIST, ASA, ANNICA, KRISTINA;SAMUELSSON, BENGT, BERTIL;VENDEVILLE, SANDRINE, MARIE HELENE 发明人 ANTONOV, DMITRY;NILSSON, KARL, MAGNUS;RABOISSON, PIERRE JEAN-MARIE BERNARD;ROSENQUIST, ASA, ANNICA, KRISTINA;SAMUELSSON, BENGT, BERTIL;VENDEVILLE, SANDRINE, MARIE HELENE
分类号 C07F9/6561;A61K31/675;A61P31/14 主分类号 C07F9/6561
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