发明名称 GLYT1 TRANSPORTER INHIBITORS AND USES THEREOF IN TREATMENT OF NEUROLOGICAL AND NEUROPSYCHIATRIC DISORDERS
摘要 <p>Compounds of formula (I) or a salt thereof are provided: wherein R&lt;SUP&gt;6&lt;/SUP&gt;, R&lt;SUP&gt;7&lt;/SUP&gt;, R&lt;SUP&gt;9&lt;/SUP&gt;, R&lt;SUP&gt;10&lt;/SUP&gt;, R&lt;SUP&gt;11&lt;/SUP&gt;, X, n, p, Ar and m are as defined in the description. Uses of the compounds as medicaments, and in the manufacture of medicament for treating neurological and neuropsychiatric disorders, in particular psychoses, dementia or attention deficit disorder are also disclosed. The invention further discloses pharmaceutical compositions and combinations comprising the compounds.</p>
申请公布号 WO2008092876(A1) 申请公布日期 2008.08.07
申请号 WO2008EP51082 申请日期 2008.01.30
申请人 GLAXO GROUP LIMITED;UNIVERSITY OF NOTTINGHAM;AHMAD, NADIA, MAMOONA;LAI, JUSTINE, YEUN QUAI;ANDREOTTI, DANIELE;MARSHALL, HOWARD, ROBERT;NASH, DAVID, JOHN;PORTER, RODERICK, ALAN 发明人 AHMAD, NADIA, MAMOONA;LAI, JUSTINE, YEUN QUAI;ANDREOTTI, DANIELE;MARSHALL, HOWARD, ROBERT;NASH, DAVID, JOHN;PORTER, RODERICK, ALAN
分类号 C07D471/10;A61K31/438;A61P25/00;A61P25/18;A61P25/28 主分类号 C07D471/10
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