发明名称 |
8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
摘要 |
The present invention relates to substituted xanthines of general formula wherein R<SUP>1 </SUP>to R<SUP>3 </SUP>are defined as in claims 1 to 16 , the tautomers, the stereoisomers, the mixtures, the prodrugs thereof and the salts thereof which have valuable pharmacological properties, particularly an inhibiting effect on the activity of the enzyme dipeptidylpeptidase-IV (DPP-IV).
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申请公布号 |
US7407955(B2) |
申请公布日期 |
2008.08.05 |
申请号 |
US20030639036 |
申请日期 |
2003.08.12 |
申请人 |
BOEHRINGER INGELHEIM PHARMA GMBH & CO., KG |
发明人 |
HIMMELSBACH FRANK;LANGKOPF ELKE;ECKHARDT MATTHIAS;MARK MICHAEL;MAIER ROLAND;LOTZ RALF R. H.;TADAYYON MOHAMMAD |
分类号 |
C07D473/06;A61K31/52;A61P3/04;A61P3/10;A61P19/02;C07D473/04;C07D473/08;C07D519/00 |
主分类号 |
C07D473/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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