| 发明名称 |
N3-HETEROARYL SUBSTITUTED TRIAZOLES AND N5-HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS |
| 摘要 |
N<SUP>3</SUP>-Heteroaryl substituted triazoles and N<SUP>5</SUP>-heteroaryl substituted triazoles and pharmaceutical compositions containing the compounds are disclosed as being useful in inhibiting the activity of the receptor protein tyrosine kinase Axl. Methods of using the compounds in treating diseases or conditions associated with Axl activity are also disclosed.
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| 申请公布号 |
US2008182862(A1) |
申请公布日期 |
2008.07.31 |
| 申请号 |
US20070966894 |
申请日期 |
2007.12.28 |
| 申请人 |
RIGEL PHARMACEUTICALS, INC. |
发明人 |
DING PINGYU;GOFF DANE;ZHANG JING;SINGH RAJINDER;HOLLAND SACHA;YU JIAXIN;HECKRODT THILO J.;LITVAK JOANE |
| 分类号 |
A61K31/4985;A61K31/4196;A61K31/498;C07D249/14;C07D403/02;C07D495/04 |
主分类号 |
A61K31/4985 |
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