| 发明名称 |
2-(PIPERIDIN-4-YL)-4-PHENOXY- OR PHENYLAMINO-PYRIMIDINE DERIVATIVES AS NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS |
| 摘要 |
The present invention provides for compounds useful for treating an HIV infection, or preventing an HIV infection, or treating AIDS or ARC. The compounds of the invention are of formula (I) wherein R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>5a</SUP>, R<SUP>5b</SUP>, R<SUP>6a</SUP>, R<SUP>6b</SUP> and X are as herein defined. Also disclosed in the present invention are methods of treating an HIV infection with compounds defined herein and pharmaceutical compositions containing said compounds. |
| 申请公布号 |
WO2008071587(A3) |
申请公布日期 |
2008.07.31 |
| 申请号 |
WO2007EP63224 |
申请日期 |
2007.12.04 |
| 申请人 |
F. HOFFMANN-LA ROCHE AG;BROTHERTON-PLEISS, CHRISTINE, E.;KERTESZ, DENIS, JOHN;YANG, MINMIN |
发明人 |
BROTHERTON-PLEISS, CHRISTINE, E.;KERTESZ, DENIS, JOHN;YANG, MINMIN |
| 分类号 |
C07D403/12;A61K31/502;A61P31/18;C07D401/14;C07D403/14;C07D471/10 |
主分类号 |
C07D403/12 |
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