发明名称 |
PROCESS OF MAKING SUBSTITUTED PYRAZOLES |
摘要 |
Disclosed is a process of making substituted pyrazoles (I) from substituted benzophenone hydrazones (II) with a variety of 1,3-bifunctional substrates (III) under acid conditions. The pyrazole compounds are useful for making pharmaceutical compounds. In said formula, wherein X is chosen from -CN and - C(O)-R3 wherein if X is CN then R3 in the product formula (I) is amino.
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申请公布号 |
CA2387762(C) |
申请公布日期 |
2008.07.29 |
申请号 |
CA20002387762 |
申请日期 |
2000.10.27 |
申请人 |
BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. |
发明人 |
BARON, JAMES A.;FARINA, VITTORIO;HADDAD, NIZAR |
分类号 |
C07D231/12;A61K31/415;A61P9/10;A61P43/00;C07B61/00;C07D231/38;C07D401/04 |
主分类号 |
C07D231/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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