USE OF I) A POLYGLYCOL AND N) AN ACTIVE DRUG SUBSTANCE FOR THE PREPARATION OF A PHARMACEUTICAL COMPOSITION FOR I) MITIGATING THE RISK OF ALCOHOL INDUCED DOSE DUMPING AND/OR II) REDUCING THE RISK OF DRUG ABUSE
摘要
<p>Abuse resistant polyglycol-based pharmaceutical compositions are disclosed. The composition contains one or more polyglycols and one or more active substances and it is resistant to crushing, melting and/or extraction. Moreover, such compositions have the same or lower solubility in ethanolic-aqueous medium, i.e. they are not subject to ethanol-induced dose dumping effect.</p>
申请公布号
WO2008086804(A2)
申请公布日期
2008.07.24
申请号
WO2008DK00016
申请日期
2008.01.16
申请人
EGALET A/S;DOWNIE, KEN;PEDERSEN, ANDERS VAGNOE;HAAHR, ANNE-METTE;HEMMINGSEN, PERNILLE HOEYRUP;BAR-SHALOM, DANIEL
发明人
DOWNIE, KEN;PEDERSEN, ANDERS VAGNOE;HAAHR, ANNE-METTE;HEMMINGSEN, PERNILLE HOEYRUP;BAR-SHALOM, DANIEL