发明名称 RAPAMYCIN (MACROLIDE) SEMI-SYNTHETIC ANALOGUE IMMUNOMODULATOR
摘要 PROBLEM TO BE SOLVED: To provide a new macrolide compound, to provide a rapamycin semi-synthetic analogue, and to provide their pharmaceutically acceptable salts, esters, amides and prodrugs. SOLUTION: A method for producing the compound represented by formula (IV), an intermediate useful for the method, a medicine composition, and a method for treating immunomodulation diseases are provided. COPYRIGHT: (C)2008,JPO&INPIT
申请公布号 JP2008150391(A) 申请公布日期 2008.07.03
申请号 JP20080025066 申请日期 2008.02.05
申请人 ABBOTT LAB 发明人 OR YAT SUN;LULY JAY R;WAGNER ROLF
分类号 C07D498/18;A61K31/439;A61K31/444;A61K31/4545;A61K31/496;A61K31/5377;A61P37/02 主分类号 C07D498/18
代理机构 代理人
主权项
地址