发明名称 |
PROCESSES FOR PREPARING (R)-8-CHLORO-1-METHYL-2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINE AND INTERMEDIATES THEREOF |
摘要 |
The present invention provides processes and intermediates for the prepar ation of (R)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine and salts thereof which are useful as serotonin-2C (5-HT2C) receptor agonists for the treatment of, for example, obesity.
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申请公布号 |
CA2670285(A1) |
申请公布日期 |
2008.06.12 |
申请号 |
CA20072670285 |
申请日期 |
2007.12.04 |
申请人 |
ARENA PHARMACEUTICALS, INC. |
发明人 |
FRITCH, JOHN ROBERT;CARLOS, MARLON;MA, YOU-AN;GHARBAOUI, TAWFIK;TANDEL, SAGUN K. |
分类号 |
C07C231/02;C07C233/22;C07D223/16;C07D263/10 |
主分类号 |
C07C231/02 |
代理机构 |
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地址 |
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