发明名称 Diaryl ethers as opioid receptor antagonist
摘要 A compound of the formula (I) wherein the variables X<SUB>1 </SUB>to X<SUB>10</SUB>, R<SUP>1 </SUP>to R<SUP>7 </SUP>including R<SUP>3'</SUP>, E, v, y, z, A and B are as described, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixtures thereof, useful for the treatment, prevention or amelioration of obesity and Related Diseases is disclosed
申请公布号 US7381719(B2) 申请公布日期 2008.06.03
申请号 US20050526960 申请日期 2005.03.03
申请人 ELI LILLY AND COMPANY 发明人 BLANCO-PILLADO MARIA-JESUS;DE LA TORRE MARTA GARCIA;DIAZ BUEZO NURIA;HOLLOWAY WILLIAM GLEN;MATT JAMES EDWARD;MITCH CHARLES HOWARD;PEDREGAL-TERCERO CONCEPCION;SMITH DANA RAE;STUCKY RUSSELL DEAN;TAKEUCHI KUMIKO
分类号 A61K31/54;A61K31/4965;A61K31/497;A61K31/50;A61K31/535;A61P3/04;C07C235/46;C07D213/38;C07D213/64;C07D213/643;C07D213/78;C07D213/81;C07D213/82;C07D217/04;C07D237/24;C07D241/02;C07D241/24;C07D307/14;C07D333/20;C07D401/00;C07D401/06;C07D401/12;C07D401/14;C07D403/00;C07D405/00;C07D405/12;C07D409/00;C07D409/12;C07D409/14;C07D411/00;C07D413/00;C07D413/12;C07D417/00;C07D417/12;C07D417/14;C07D419/00 主分类号 A61K31/54
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