发明名称 |
FORMA CRISTALINA DE 4-(2-(4,4-DIMETIL-2-OXOOXAZOLIDIN-3-IL)TRIAZOL-4-IL)BENZONITRILO; METODO DE PREPARACION; COMPOSICION FARMACEUTICA; KIT FARMACEUTICO; Y USO PARA TRATAR SINDROME DE OVARIO POLIQUISTICO, CANCER, ENTRE OTRAS ENFERMEDADES. |
摘要 |
A polymorph Form II of 4-(2-(4,4-dimethyl-2-oxooxazolidin-3-yl)thiazol-4-yl)benzonitrile and methods of preparing Form II are described. Also provided are methods of contraception, treating or preventing fibroids, uterine leiomyomata, endometriosis, dysfunctional bleeding, polycystic ovary syndrome, and hormone-dependent carcinomas, providing hormone replacement therapy, stimulating food intake, and synchronizing estrus including using polymorph Form II of 4-(2-(4,4-dimethyl-2-oxooxazolidin-3-yl)thiazol-4-yl)benzonitrile. Further provided are methods for preparing polymorph Form I of 4-(2-(4,4-dimethyl-2-oxooxazolidin-3-yl)thiazol-4-yl)benzonitrile from polymorph Form II of 4-(2-(4,4-dimethyl-2-oxooxazolidin-3-yl)thiazol-4-yl)benzonitrile. |
申请公布号 |
CL2008000663(A1) |
申请公布日期 |
2008.05.30 |
申请号 |
CL20080000663 |
申请日期 |
2008.03.06 |
申请人 |
WYETH |
发明人 |
MIRMEHRABI, MAHNOUD, NIU, YUPING, TADAYON, ABDOLSAMAD, DESHMUKH, SUBODH, KU, M. SHERRY. |
分类号 |
A61K31/427;A61P5/00;A61P35/00;C07D417/04 |
主分类号 |
A61K31/427 |
代理机构 |
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