NOVEL INTERMEDIATES FOR THE PREPARATION OF A GLYT1 INHIBITOR
摘要
This invention relates to an improved process for preparing the glycine transport 1 (GlyT1) inhibitor (Z)-N-(1-(4-(2-furyl)phenyl)-1-(3-thienyl-prop-1-en-3-yl) sarcosine via the novel intermediate (Z)-3-(4-(2-furyl)phenyl)-3-(3-thienyl)-prop-2-en-1-ol and the preparation of the latter.
申请公布号
WO2008040669(A3)
申请公布日期
2008.05.29
申请号
WO2007EP60203
申请日期
2007.09.26
申请人
JANSSEN PHARMACEUTICA N.V.;HOUPIS, IOANNIS, NICOLAOS;SCHILS, DIDIER, PHILIPPE, ROBERT
发明人
HOUPIS, IOANNIS, NICOLAOS;SCHILS, DIDIER, PHILIPPE, ROBERT
