发明名称 |
Pyrimidine derivatives for the prevention of HIV infection |
摘要 |
This invention concerns the use of a compound for the manufacture of a medicament for the prevention of HIV infection via sexual intercourse and related intimate contact between partners, wherein the compound is a compound of formula (I) a N-oxide, a pharmaceutically acceptable addition salt, a quaternary amine and a stereochemically isomeric form thereof, wherein the ring containing -a<SUP>1</SUP>=a<SUP>2</SUP>-a<SUP>3</SUP>=a<SUP>4</SUP>- and -b<SUP>1</SUP>=b<SUP>2</SUP>-b<SUP>3</SUP>=b<SUP>4</SUP>- represents phenyl, pyridyl, pyrimidinyl, pirazinyl, pyridazinyl; and pharmaceutical compositions comprising them. |
申请公布号 |
ZA200506253(B) |
申请公布日期 |
2008.05.28 |
申请号 |
ZA20050006253 |
申请日期 |
2005.08.04 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
GUILLEMONT, JEROME EMILE GEORGES;JANSSEN, PAUL ADRIAAN JAN;LEWI, PAULUS JOANNES;KOYMANS, LUCINE MARIA HENRICUS;VINKERS, HENDRIK MAARTEN;PASQUIER, ELISABETH THERESE JEANNE;HEERES, JAN;DE JONGE, MARC RENE;DAEYAERT, FREDERIK FRANS DESIRE |
分类号 |
A61K;A61P;A61P31/18;C07D;C07D239/46 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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