发明名称 |
BENZENE DERIVATIVE OR SALT THEREOF |
摘要 |
[PROBLEMS] To provide a compound which has an anticoagulation activity based on the inhibition of an activated blood coagulation factor X and is useful as a blood coagulation inhibitor or a preventive or therapeutic agent for a disease caused by thrombus or embolus. [MEANS FOR SOLVING PROBLEMS] A benzene derivative characterized by having a chemical structure in which a phenol ring and a benzene ring are bound via an amide bond and the phenol ring is further bound to a benzene ring or a heteroaryl ring via an amide bond or a salt thereof. These comounds have an excellent activated blood coagulation factor X inhibitory action and particularly has an excellent oral activity.
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申请公布号 |
KR20080046711(A) |
申请公布日期 |
2008.05.27 |
申请号 |
KR20087008720 |
申请日期 |
2008.04.11 |
申请人 |
ASTELLAS PHARMA INC. |
发明人 |
HIRAYAMA FUKUSHI;FUJIYASU JIRO;KAGA DAISUKE;NEGORO KENJI;SASUGA DAISUKE;SEKI NORIO;SUZUKI KEN ICHI |
分类号 |
C07D211/74;A61K31/435;C07D213/64;C07D413/14 |
主分类号 |
C07D211/74 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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