摘要 |
<p>Disclosed is a method for producing a 2-alkyl-3-aminothiophene derivative represented by the general formula (2) below by reducing a 2-alkenyl-3-aminothiophene derivative represented by one of the general formulae (1a)-(1d) below, a mixture thereof or a salt thereof without using a protecting group. (In the formulae, R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP> and R<SUP>4</SUP> independently represent a hydrogen atom, an alkyl group having 1-12 carbon atoms or the like; and R<SUP>5</SUP> and R<SUP>6</SUP> independently represent a hydrogen atom, a halogen atom, an alkyl group having 1-12 carbon atoms or the like.) This method enables to commercially produce a 2-alkyl-3-aminothiophene derivative which is useful as an agricultural chemical intermediate at low cost without using an economically disadvantageous protecting group for an amino group.</p> |
申请人 |
MITSUI CHEMICALS, INC.;KAKIMOTO, TAKESHI;AOKI, YOJI;URA, DAISUKE;ENOMOTO, MIKI;KAMEKAWA, HISATO;KITASHIMA, TOSHIO |
发明人 |
KAKIMOTO, TAKESHI;AOKI, YOJI;URA, DAISUKE;ENOMOTO, MIKI;KAMEKAWA, HISATO;KITASHIMA, TOSHIO |