发明名称 TRIAZOLOPYRIMIDINE DERIVATIVES AS ADP P2Y12 RECEPTOR ANTAGONISTS
摘要 <p>The present invention is directed to novel bicyclic triazolopyrimidine compounds of Formula (I) or a form thereof, wherein X&lt;SUB&gt;1&lt;/SUB&gt;, X&lt;SUB&gt;2&lt;/SUB&gt;, R&lt;SUB&gt;1&lt;/SUB&gt; R&lt;SUB&gt;2&lt;/SUB&gt;, R&lt;SUB&gt;3&lt;/SUB&gt; and R&lt;SUB&gt;4&lt;/SUB&gt; are as defined herein, and their methods of preparation and use as ADP inhibitors.</p>
申请公布号 WO2008054796(A2) 申请公布日期 2008.05.08
申请号 WO2007US23016 申请日期 2007.10.31
申请人 YE, HONG;JANSSEN PHARMACEUTICA, N.V.;ZHANG, HAN-CHENG;MARYANOFF, BRUCE, E.;CHEN, CAILIN 发明人 ZHANG, HAN-CHENG;MARYANOFF, BRUCE, E.;YE, HONG;CHEN, CAILIN
分类号 A61K31/519 主分类号 A61K31/519
代理机构 代理人
主权项
地址