发明名称 |
TRIAZABENZO(E)AZULENE DERIVATIVES FOR THE TREATMENT OF TUMOURS |
摘要 |
Novel triaza-benzo[e]azulene derivatives of the formula (I) in which R1, R2 and R3 are each as defined in claim 1 are inhibitors of TGF-beta receptor kinase, and can be used, inter alia, for the treatment of tumors.
|
申请公布号 |
CA2668562(A1) |
申请公布日期 |
2008.05.08 |
申请号 |
CA20072668562 |
申请日期 |
2007.09.29 |
申请人 |
MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG |
发明人 |
AMENDT, CHRISTIANE;GREINER, HARTMUT;HOELZEMANN, GUENTER |
分类号 |
C07D487/04;A61K31/55;A61P35/00 |
主分类号 |
C07D487/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|