发明名称 |
Benzoxazole Carboxamides For Treating CINV and IBS-D |
摘要 |
Compounds of formulae I and II: are disclosed as 5-HT<SUB>3 </SUB>inhibitors. Those compounds that exhibit central activity are useful in treating CINV; those that inhibit peripheral receptors are useful to treat IBS-D.
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申请公布号 |
US2008108609(A1) |
申请公布日期 |
2008.05.08 |
申请号 |
US20070934523 |
申请日期 |
2007.11.02 |
申请人 |
AMR TECHNOLOGY, INC. |
发明人 |
FAIRFAX DAVID J.;YANG ZHICAI |
分类号 |
C07D263/56;A61K31/423;A61K31/4375;A61K31/439;A61K31/443;A61K31/4523;A61K31/496;A61K31/5377;A61P1/00;C07D401/14;C07D413/00;C07D453/00 |
主分类号 |
C07D263/56 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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