发明名称 Benzoxazole Carboxamides For Treating CINV and IBS-D
摘要 Compounds of formulae I and II: are disclosed as 5-HT<SUB>3 </SUB>inhibitors. Those compounds that exhibit central activity are useful in treating CINV; those that inhibit peripheral receptors are useful to treat IBS-D.
申请公布号 US2008108609(A1) 申请公布日期 2008.05.08
申请号 US20070934523 申请日期 2007.11.02
申请人 AMR TECHNOLOGY, INC. 发明人 FAIRFAX DAVID J.;YANG ZHICAI
分类号 C07D263/56;A61K31/423;A61K31/4375;A61K31/439;A61K31/443;A61K31/4523;A61K31/496;A61K31/5377;A61P1/00;C07D401/14;C07D413/00;C07D453/00 主分类号 C07D263/56
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