发明名称 THIAZOLE DERIVATIVE
摘要 [PROBLEMS] To provide a compound which is useful as a GK activator. [MEANS FOR SOLVING PROBLEMS] As a result of an extensive study on thiazole derivatives, it is found that a compound having an oxamoyl group, a glycol group or the like on a thiazole ring and a compound having an acetamide group substituted by a dicyclic heteroaryl group such as a quinolyl have a good GK activation effect. These compounds are useful as therapeutic agents for diabetes, particularly type 2 diabetes.
申请公布号 KR20080040046(A) 申请公布日期 2008.05.07
申请号 KR20087007622 申请日期 2008.03.28
申请人 ASTELLAS PHARMA INC. 发明人 HAYAKAWA MASAHIKO;NIGAWARA TAKAHIRO;TSUCHIYA KAZUYUKI;ISHIBASHI NAOKI;OKUMURA MITSUAKI;KAWAMOTO YUICHIRO;NAGAYOSHI AKIRA
分类号 C07D277/20;A61K31/426;A61P3/10;C07D277/56 主分类号 C07D277/20
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