发明名称 BENZODIOXANE DERIVATIVES AND USES THEREOF
摘要 <p>Compounds are described herein which are agonists or partial agonists of the 2C subtype of brain serotonin receptors. The compounds have the formula I: or pharmaceutically acceptable salts thereof, wherein each of A, R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, R&lt;SUP&gt;4&lt;/SUP&gt;, R&lt;SUP&gt;a&lt;/SUP&gt;, R&lt;SUP&gt;b&lt;/SUP&gt;, R&lt;SUP&gt;c&lt;/SUP&gt;, R&lt;SUP&gt;d&lt;/SUP&gt;, R&lt;SUP&gt;e&lt;/SUP&gt;, R&lt;SUP&gt;x&lt;/SUP&gt;, R&lt;SUP&gt;y&lt;/SUP&gt;, m, n and each == group are as defined herein. Such compounds, and compositions thereof, are useful for treating a variety of central nervous system disorders such as schizophrenia.</p>
申请公布号 WO2008052086(A1) 申请公布日期 2008.05.02
申请号 WO2007US82450 申请日期 2007.10.24
申请人 WYETH;STACK, GARY, PAUL;DEMAIO, WILLIAM;ERVE, JOHN, CHUCK, LEM;VISHWANATHAN, KARTHICK;WANG, JIANYAO;VASHISHTHA, SARVESH 发明人 STACK, GARY, PAUL;DEMAIO, WILLIAM;ERVE, JOHN, CHUCK, LEM;VISHWANATHAN, KARTHICK;WANG, JIANYAO;VASHISHTHA, SARVESH
分类号 C07D319/20;A61K31/357;A61P25/18 主分类号 C07D319/20
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