A chemical genus of purines, which are useful as PKC.theta. inhibitors, i s disclosed. The genus is represented by the formula (I); A representative e xample is: (II)
申请公布号
CA2666940(A1)
申请公布日期
2008.05.02
申请号
CA20072666940
申请日期
2007.10.19
申请人
N.V. ORGANON;PHARMACOPEIA, L.L.C.
发明人
WIJKMANS, JACOBUS CORNELIS HENRICUS MARIA;KINGSBURY, CELIA;TEERHUIS, NEELTJE MIRANDA;OHLMEYER, MICHAEL;DILLER, DAVID;HO, KOC-KAN;CHAN, JUI HSIANG;ROUGHTON, ANDREW;LOMMERSE, JOHANNES PETRUS MARIA;NEAGU, IRINA