发明名称 |
GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF |
摘要 |
COMPOUNDS OF FORMULA (1) WHEREIN R1, R2, R3, R4, R5, R6, AND X ARE AS DEFINED HEREIN FOR FORMULA (1A) AND FORMULA (IB, OR A TAUTOMER, PRODRUG, SOLVATE, OR SALT THEREOF; PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDS, AND METHODS OF MODULATING THE GLUCOCORTICOID RECEPTOR FUNCTION AND METHODS OF TREATING DISEASE-STATES OR CONDITIONS MEDIATED BY THE GLUCOCORTICOID RECEPTOR FUNCTION OR CHARACTERIZED BY INFLAMMATORY, ALLERGIC, OR PROLIFERATIVE PROCESSES IN A PATIENT USING THESE COMPOUNDS.
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申请公布号 |
MY135423(A) |
申请公布日期 |
2008.04.30 |
申请号 |
MYPI20040009 |
申请日期 |
2004.01.02 |
申请人 |
BOEHRINGER INGELHEIM PHARMACEUTICALS, INC |
发明人 |
JOHN R. PROUDFOOT;JOHN ROBINSON REGAN;DAVID S. THOMSON;DANIEL KUZMICH;THOMAS WAI-HO LEE;THOMAS MARTIN KIRRANE,JR |
分类号 |
C07D207/14;C07D209/08;C07D209/34;C07D209/44;C07D209/48;C07D211/14;C07D211/18;C07D211/46;C07D211/58;C07D211/60;C07D211/62;C07D211/74;C07D213/64;C07D213/68;C07D213/69;C07D213/74;C07D213/85;C07D215/06;C07D215/22;C07D215/227;C07D215/233;C07D215/42;C07D217/04;C07D231/56;C07D237/28;C07D239/42;C07D239/88;C07D239/90;C07D241/04;C07D241/08;C07D241/38;C07D241/42;C07D241/44;C07D243/08;C07D243/14;C07D265/22;C07D265/36;C07D279/12;C07D279/16;C07D295/084;C07D295/112;C07D295/15;C07D295/185;C07D295/205;C07D307/24;C07D307/68;C07D317/58;C07D401/04;C07D401/06;C07D401/10;C07D401/14;C07D405/06;C07D405/10;C07D409/06;C07D409/10;C07D413/06;C07D413/10;C07D417/06;C07D471/04;C07D487/08 |
主分类号 |
C07D207/14 |
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