发明名称 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS FOR USE AS STEAROYL COA DESATURASE INHIBITORS
摘要 The present invention discloses bicyclic nitrogen-containing heterocyclic compounds for use as inhibitors of stearoyl-CoA desaturase. The compounds are useful in treating and/or preventing various human diseases, mediated by stearoyl-CoA desaturase (SCD) enzymes, especially diseases related to abnormal lipid levels, cardiovascular disease, diabetes, obesity, oily skin conditions, metabolic syndrome, and the like.
申请公布号 WO2008043087(A2) 申请公布日期 2008.04.10
申请号 WO2007US80627 申请日期 2007.10.05
申请人 CV THERAPEUTICS, INC.;ZABLOCKI, JEFF;GLUSHKOV, AUDREY;ZILBERSHTEIN, TIMUR;PARKHILL, ERIC;KOLTUN, DMITRY;VASILEVICH, NATALYA;CHISHOLM, JEFFREY;IVANOV, ALEXEY 发明人 ZABLOCKI, JEFF;GLUSHKOV, AUDREY;ZILBERSHTEIN, TIMUR;PARKHILL, ERIC;KOLTUN, DMITRY;VASILEVICH, NATALYA;CHISHOLM, JEFFREY;IVANOV, ALEXEY
分类号 C07D241/44;A61K31/519;A61P35/00;C07D401/04;C07D471/04 主分类号 C07D241/44
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