发明名称 Purinones and 1H-imidazopyridinones as PKC-theta inhibitors
摘要 A chemical genus of purinones and 1H-imidazopyridinones, which are useful as PKCtheta inhibitors, and their methods of use are disclosed. The genus is represented by the formula I: A representative example is:
申请公布号 US2008085909(A1) 申请公布日期 2008.04.10
申请号 US20070701632 申请日期 2007.02.02
申请人 PHARMACOPEIA DRUG DISCOVERY, INC. 发明人 ROUGHTON ANDREW;RONG YAJING;HO KOC KAN;OHLMEYER MICHAEL;DILLER DAVID
分类号 A61K31/522;A61P3/10;A61P11/06;A61P29/00;A61P35/00;A61P37/00;C07D473/18 主分类号 A61K31/522
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