PIPERIDINE AND PIPERAZINE DERIVATIVES AS P2X3 ANTAGONISTS
摘要
Compounds of formula (I) wherein R1, R2a, R2b, R3, Y, X, A, R6, R7 and R8 are as described herein, are modulators of P2X3 useful for the treatment of pain and genitourinary, gastrointestinal, and respiratory disorders. ® KIPO & WIPO 2008
申请公布号
KR20080027943(A)
申请公布日期
2008.03.28
申请号
KR20087003538
申请日期
2006.08.03
申请人
F. HOFFMANN-LA ROCHE AG
发明人
BROTHERTON PLEISS CHRISTINE E.;DILLON MICHAEL PATRICK;GLEASON SHELLEY K.;LIN CLARA JEOU JEN;SCHOENFELD RYAN CRAIG;VILLA MARZIA;ZHAI YANSHENG