发明名称 PYRAZOLONE DERIVATIVE AND PDE INHIBITING AGENT CONTAINING THE DERIVATIVE AS ACTIVE COMPONENT
摘要 PROBLEM TO BE SOLVED: To provide a new pyrazolone derivative useful as a medicine having phosphodiesterase inhibiting action. SOLUTION: The pyrazolone derivative is expressed by general formula (1) (a concrete example of the derivative is 3-(2-ethyl-8-methoxyquinolin-5-yl)-4,4-dimethyl-1H-pyrazol-5(4H)-one). COPYRIGHT: (C)2008,JPO&INPIT
申请公布号 JP2008069144(A) 申请公布日期 2008.03.27
申请号 JP20070212079 申请日期 2007.08.16
申请人 KYORIN PHARMACEUT CO LTD 发明人 KONO YASUSHI;TAKITA TETSUSHI;OCHIAI KOJI;EIRAKU TOMOHIKO;KOJIMA AKIHIKO
分类号 C07D401/04;A61K31/4155;A61K31/4184;A61K31/428;A61K31/437;A61K31/4709;A61P1/04;A61P3/00;A61P3/04;A61P7/02;A61P9/04;A61P9/10;A61P9/12;A61P11/00;A61P11/02;A61P11/06;A61P15/10;A61P17/00;A61P19/02;A61P25/00;A61P25/14;A61P25/16;A61P25/18;A61P25/24;A61P25/28;A61P29/00;A61P37/08;A61P43/00;C07D403/04;C07D405/04;C07D409/04;C07D417/04;C07D471/04 主分类号 C07D401/04
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