INDOLYLALKYLPYRIDIN-2-AMINES FOR THE INHIBITION OF BETA-SECRETASE
摘要
INDOLYLALKYLPYRIDIN-2-AMINES FOR THE INHIBITION OF ß-SECRETASE The present invention provides an indolylalkylpyridin-2-amine compound of formula I CHEMICAL FORMULA SHOULD BE INSERTED HERE AS IT APPEARS ON THE ABSTRACT IN PAPER FORM. The present invention also provides methods for the use thereof to inhibit ß-secretase (BACE) and treat ß-amyloid deposits and neurofibrillary tangles.
申请公布号
WO2008036196(A2)
申请公布日期
2008.03.27
申请号
WO2007US19945
申请日期
2007.09.14
申请人
WYETH;YAN, YINFA;ZHOU, PING;FAN, YI;ROBICHAUD, ALBERT JEAN;MALAMAS, MICHAEL SOTIRIOS
发明人
YAN, YINFA;ZHOU, PING;FAN, YI;ROBICHAUD, ALBERT JEAN;MALAMAS, MICHAEL SOTIRIOS