A process for making anastrozole using a 1-substituted triazole can reduce formation of the undesired iso-anastrozole. A typical process is represented by (I), wherein compound (10) is a 1-substituted triazole and compound (1) is anastrozole.
申请公布号
WO2008034644(A2)
申请公布日期
2008.03.27
申请号
WO2007EP08338
申请日期
2007.09.20
申请人
SYNTHON B.V.;BENES, MICHAL;PROSEK, ZDENEK;HYKL, JIRI;PIS, JAROSLAV
发明人
BENES, MICHAL;PROSEK, ZDENEK;HYKL, JIRI;PIS, JAROSLAV
