发明名称 METHOD FOR PRODUCING NEBIVOLOL
摘要 The invention relates to a method for producing the racemic active ingredient Nebivolol, according to which diastereomer cyanhydrins are produced and separated, and the separated diastereomers are coupled together following a transformation, preferably a partial or full reduction of the cyano group or a Pinner saponification. ® KIPO & WIPO 2008
申请公布号 KR20080027368(A) 申请公布日期 2008.03.26
申请号 KR20087001837 申请日期 2008.01.23
申请人 PHARMACON - FORSCHUNG UND BERATUNG GMBH 发明人 NOE CHRISTIAN R.;JASIC MUHAMED;KOLLMANN HERMANN;LACHMANN BODO
分类号 C07D407/12 主分类号 C07D407/12
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