发明名称 NOVEL ARYLAMINO N-HETERARYLS AS MEK INHIBITORS
摘要 The invention provides novel arylamino N-heteroaryl MEK inhibitors of Formula (I): Such compounds are MEK inhibitors that are useful in the treatment of hyperproliferative diseases, such as cancer and inflammation. Also disclosed. is the treatment of a hyperproliferative disease in mammals, and pharmaceutical compositions containing such compounds.
申请公布号 WO2007123939(A8) 申请公布日期 2008.03.13
申请号 WO2007US09461 申请日期 2007.04.18
申请人 APPLIED RESEARCH SYSTEMS ARS HOLDING N.V.;GOUTOPOULOS, ANDREAS;ASKEW, JR., BENNY, C.;DIEP, NHUT, KIET;KARRA, SRINIVASA;SCHWARZ, MATTHIAS;YU, HENRY 发明人 GOUTOPOULOS, ANDREAS;ASKEW, JR., BENNY, C.;DIEP, NHUT, KIET;KARRA, SRINIVASA;SCHWARZ, MATTHIAS;YU, HENRY
分类号 C07D213/79;A61K31/44;A61K31/50;A61P29/00;A61P35/00;C07D213/80;C07D213/81;C07D213/82;C07D213/84;C07D237/24;C07D405/12 主分类号 C07D213/79
代理机构 代理人
主权项
地址